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Table 1 Effect of tested compounds on hERG current density at +20 mV (I +20 )

From: Mitigating prolonged QT interval in cancer nanodrug development for accelerated clinical translation

Compound tested

Statistically significant inhibition starting at (μM)

Maximal inhibition (%)

Statistically significant reversibility of the Washout

Calculated IC50 (μM)

Voltage dependence

HNC-NP

18

24.8

No

n/a

Yes

HNC-PS

6

40.2

No

n/a

Yes

HNC-PS-C

6

25.2

No

n/a

Yes

Curcumin

12

77.8

No

8.5

Yes

Liposomal curcumin

6 only

30

No

n/a

No