From: Engineering of small-molecule lipidic prodrugs as novel nanomedicines for enhanced drug delivery
Properties | Lipids | Drugs | Refs. |
---|---|---|---|
High drug loading | Oleic acid/linoleic acid/stearic acid/phospholipid | Docetaxel/paclitaxel/5-fluorouracil | |
High intracellular uptake and cytotoxicity | Linoleic acid/palmityl/palmitic acid/linolenic acid | Gemcitabine/doxorubicin | |
Enhancing the performance of oral administration | Undecanoate/triglyceride/oleic acid/taurocholic acid/deoxycholic acid | 7-Ethyl-10-hydroxycamptothecin/mycophenolic acid/docetaxel/heparin | |
Increasing the antitumor efficacy with low systemic toxicity | Docosahexaenoic acid/oleic acid/linolenic acid/phospholipid | Paclitaxel/cabazitaxel/porphyrin |